Tuesday, October 11, 2016

Chloramphenicol Eye Drops BP 0.5% W / V





1. Name Of The Medicinal Product



Chloramphenicol Eye Drops BP 0.5% W/V


2. Qualitative And Quantitative Composition







Active ingredient:




Chloramphenicol




0.5g IN 100ml



3. Pharmaceutical Form



Eye Drops



4. Clinical Particulars



4.1 Therapeutic Indications



Treatment of bacterial conjunctivitis caused by the organisms Escherichia coli, Haemophilus influenzae, Staphylococcus aureus, Streptococcus haemolyticus, Morax-Axenfield and others



4.2 Posology And Method Of Administration



The recommended dosage for adults, children and infants of all age groups is two drops to be applied to the affected eye every three hours or more frequently if required. Treatment should be continued for at least 48 hours after eye appears normal.



4.3 Contraindications



• Hypersensitivity to chloramphenicol or to any other ingredient of the drops.



• Myelosuppression during previous exposure to chloramphenicol.



• Family history of dyscrasias.



4.4 Special Warnings And Precautions For Use



Chloramphenicol is absorbed systemically from the eye and toxicity has been reported following chronic exposure.



Bone marrow hypoplasia, including aplastic anaemia and death, has been reported following topical use of chloramphenicol. Whilst the hazard is a rare one, it should be borne in mind when assessing the benefits expected from the use of the compound.



Where chloramphenicol eye drops are used on a long term or intermittent basis, it may be advisable to perform a routine blood profile before therapy and at appropriate intervals thereafter to detect any haemopoietic abnormalities.



In severe infections the topical use of chloramphenicol should be supplemented by appropriate systemic treatment. The prolonged use of antibiotics may occasionally result in overgrowth of non susceptable organisms, including fungi. If any new infection appears during the treatment, the antibiotic should be discontinued and appropriate measures taken. Chloramphenicol should be reserved for use only for infections for which it is specifically indicated.



Soft contact lenses should not be worn during treatment with chloramphenicol eye drops due to absorption of the preservative onto the lens which may cause damage to the lens. It is recommended that all types of contact lenses be avoided during ocular infections.



Chloramphenicol Eye Drops do not provide adequate coverage against Pseudomonas aeruginosa and Serratia marcescens.



4.5 Interaction With Other Medicinal Products And Other Forms Of Interaction



Bone marrow suppressant drugs.



4.6 Pregnancy And Lactation



Safety for use in pregnancy and lactation has not been established. Therefore, use only when considered essential by the physician.



4.7 Effects On Ability To Drive And Use Machines



Transient blurring of vision may occur immediately after use and driving or using machinery should not occur until the vision is clear.



4.8 Undesirable Effects



Eye disorders:



Transient irritation, burning, stinging and sensitivity reactions such as itching and dermatitis.



Immune System Disorders:



Hypersensitivity reactions including angioedema, anaphylaxis, urticaria, fever, vesicular and maculopapular dermatitis.



Blood and lymphatic system disorders:



Bone marrow depression and rarely aplastic anaemia has been reported following topical use of chloramphenicol. Whilst the hazard is a rare one, it should be borne in mind when assessing the benefits expected from the use of this compound.



4.9 Overdose



Accidental ingestion of the drops is unlikely to cause systemic toxicity due to the low content of the antibiotic in the product. If irritation, pain, swelling, lacrimation or photophobia occur after undesired eye contact, the exposed eye(s) should be irrigated for at least 15 minutes. If symptoms persist after this, an ophthalmological examination should be considered



5. Pharmacological Properties



5.1 Pharmacodynamic Properties



Chloramphenicol is a broad spectrum antibiotic with bacteriostatic activity and is effective against a wide range of gram-negative and gram-positive organisms



5.2 Pharmacokinetic Properties



Not applicable to topical (ophthalmic) preparations.



5.3 Preclinical Safety Data



Nothing of relevance which is not included in other sections of the SPC



6. Pharmaceutical Particulars



6.1 List Of Excipients



Borax



Boric Acid



Phenyl Mercuric Nitrate



Purified Water



6.2 Incompatibilities



None known



6.3 Shelf Life








Unopened:




24 months




Opened:




28 days



6.4 Special Precautions For Storage



Protect from light.



Store between 2°C and 8°C



6.5 Nature And Contents Of Container



Low density polyethylene bottle with polystyrene spiked cap. Available in pack sizes of 5ml or 10ml



6.6 Special Precautions For Disposal And Other Handling



None



7. Marketing Authorisation Holder



FDC International Ltd



Unit 6 Fulcrum 1



Solent Way



Whiteley



Fareham



Hants PO15 7FE



United Kingdom



8. Marketing Authorisation Number(S)



PL 15872/0003



9. Date Of First Authorisation/Renewal Of The Authorisation



16 January 1998 / 07 March 2003



10. Date Of Revision Of The Text



7 October 2010





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